library.onepin.app/selank Peptide Education Library
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OnePin Peptide Library · Cognitive & Mood

Cognitive & Mood Synthetic heptapeptide Not FDA-approved · investigational Controlled substance

Selank

TP-7 · Selank Acetate

Synthetic heptapeptideTuftsin analog with Pro-Gly-Pro extensionAnxiolytic peptide (non-benzodiazepine)GABA/serotonin modulator

Selank is a synthetic heptapeptide derived from the endogenous immunomodulatory peptide tuftsin (Thr-Lys-Pro-Arg), with a stabilizing Pro-Gly-Pro C-terminal extension. Developed alongside Semax at the Institute of Molecular Genetics of the Russian Academy of Sciences, Selank is approved in Russia as a prescription anxiolytic and nootropic medication. It provides anxiolytic effects through modulation of GABAergic and serotonergic neurotransmission without the sedation, cognitive impairment, or dependence associated with benzodiazepines. Selank also enhances immune function through its tuftsin-derived immunomodulatory activity. It is commonly paired with DSIP for sleep support and with Semax for balanced nootropic effects.

Quick Start
Route
SubQ injection. Also available as nasal spray (most common in Russia).
Start low
200-500 mcg daily
Frequency
Daily, evening preferred for sleep support
Timing
No fasting required. Evening dosing preferred for sleep benefits.

Intranasal: Any time, anxiolytic effects within minutes. SubQ: Same timing. Can be paired with Semax. No fasting required.

Start here. Every protocol below is ordered lowest-first. Begin at the smallest effective dose, hold about a week to assess tolerance, and step up only if needed.

Tiered Protocols · lowest first
Quick Start
Conservative start
200-500 mcg daily · SubQ injection. Also available as nasal spray (most common in Russia). · Daily, evening preferred for sleep support
Lowest starting point. Hold about a week to assess tolerance before stepping up.
200-500 mcg daily
Daily, evening preferred for sleep support
Standard
Anxiolytic Clarity
200-500 mcg · SubQ · Daily
human study · Zozulya et al. 2001 (Bull Exp Biol Med)
200-500 mcg
Daily
Reconstitution CalculatorU-100
050100u
Draw to
units
01

How it works

Selank modulates GABA-A receptor sensitivity, enhancing inhibitory neurotransmission without directly binding the benzodiazepine site, which prevents sedation and dependence. It also influences serotonin (5-HT) metabolism by affecting tryptophan hydroxylase activity and serotonin transporter dynamics, contributing to mood stabilization and anxiety reduction. The tuftsin core (Thr-Lys-Pro-Arg) provides immunomodulatory activity by enhancing phagocytic activity of macrophages and neutrophils, natural killer cell function, and IL-6 expression. The Pro-Gly-Pro extension protects against aminopeptidase degradation, extending effective half-life. Gene expression studies show Selank modulates approximately 80 genes related to GABAergic signaling, serotonergic pathways, and immune function.

Selank modulates GABA-A receptor sensitivity, enhancing inhibitory neurotransmission without directly binding the benzodiazepine site, which prevents sedation and dependence. It also influences serotonin (5-HT) metabolism by affecting tryptophan hydroxylase activity and serotonin transporter dynamics, contributing to mood stabilization and anxiety reduction. The tuftsin core (Thr-Lys-Pro-Arg) provides immunomodulatory activity by enhancing phagocytic activity of macrophages and neutrophils, natural killer cell function, and IL-6 expression. The Pro-Gly-Pro extension protects against aminopeptidase degradation, extending effective half-life. Gene expression studies show Selank modulates approximately 80 genes related to GABAergic signaling, serotonergic pathways, and immune function.

02

What to expect

Early
Days 1–7

Days 1-3: Many users report noticeable anxiety reduction within the first few days. Sleep quality improvements if dosed in the evening. No sedation or cognitive dulling.

Mid
Weeks 2–4

Weeks 1-4: Consistent anxiolytic effects. Stress resilience improves. Sleep quality stabilizes. Immune function benefits begin to accumulate. Best results when paired with Semax for cognitive balance.

Later
Weeks 4–12

Weeks 4-8: Sustained mood and anxiety benefits. Immune modulation fully established. No tolerance or dependence develops. Cycling is recommended to maintain receptor sensitivity.

03

Evidence

HumanPresent
AnimalStrong
In-vitroPresent
2008Efficacy and possible mechanisms of action of a new peptide anxiolytic selank in the therapy of generalized anxiety disorders and neurasthenia · Zozulia AA, Neznamov GG, Siuniakov TS et al, Zhurnal Nevrologii i Psikhiatrii imeni S.S. Korsakova ↗peer reviewed
2020Functional Connectomic Approach to Studying Selank and Semax Effects · Volel B, Sysoeva O, Mershina E et al, Frontiers in Pharmacology ↗peer reviewed
2017Peptide Selank Enhances the Effect of Diazepam in Reducing Anxiety in Transgenic Mouse Lines · Volkova A, Shadrina M, Kolomin T et al, Frontiers in Pharmacology ↗peer reviewed
2016Selank Administration Affects the Expression of Some Genes Involved in GABAergic Neurotransmission · Kolomin T, Shadrina M, Slominsky P et al, Frontiers in Pharmacology ↗peer reviewed
04

The honest take

Non-benzodiazepine anxiolytic

Strongest claim. Approved in Russia for anxiety. Human studies show anxiolytic efficacy comparable to medazepam without sedation, cognitive impairment, or dependence risk.

Immune enhancement

Tuftsin-derived immunomodulatory activity is well-documented. Enhanced phagocytic activity and NK cell function. Dual anxiolytic + immune support is unique among peptides.

No tolerance or dependence
Supported

Confirmed by Russian clinical data. Selank does not bind the benzodiazepine site and does not produce tolerance, dependence, or withdrawal. Major safety advantage over benzodiazepines.

05

Interactions & stacking

What's safe to combine, and what belongs in a separate pin.

Safe & synergistic

BPC-157Non-overlapping (anxiolytic vs tissue repair)
TB-500Non-overlapping mechanisms
GHK-CuNon-overlapping mechanisms
GHKNon-overlapping mechanisms

Keep separate

CJC-1295 with DACDAC maleimide reactivity concern.
06

Side effects & safety

Commonly reported

  • Generally very well tolerated
  • Mild injection site irritation
  • Occasional mild fatigue (usually first few days)
  • Rare nasal irritation if using intranasal route

Less common & notes

  • Selank has an excellent safety profile in Russian clinical use.
  • No dependence, tolerance, or withdrawal reported.
  • No cognitive impairment.
  • Rarely, mild headache.
  • Individuals on SSRIs or other serotonergic medications should use caution as Selank modulates serotonin metabolism.
  • Consult physician if on psychiatric medications.
07

Pharmacokinetics

Illustrative plasma concentration · 24 h
Half-life
0.5h
Peak · Tmax
0.75h
Elimination
2.5h
Activity
6-12 hours (anxiolytic and GABA/serotonin modulation effects outlast plasma presence)

Storage. Store unreconstituted vials frozen (-20C) or refrigerated (2-8C). After reconstitution with BAC water, refrigerate at 2-8C. Stable for 28 days. Pro-Gly-Pro modification enhances enzymatic stability. Protect from light.

08

Regulatory status

Approved as a prescription medication in Russia for anxiety and cognitive disorders. Not FDA-approved in the United States. Available as a research peptide. WADA status: Not specifically listed. Not a controlled substance.

Put it to work

Calculate, log & track

Open Selank straight into OnePin with your vial and dose pre-filled, then let it handle the syringe math and remind you before the vial runs out.

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Go deeper

The guide & community

The complete Selank walkthrough, real protocol discussion and coaching live inside the BlessUp community on Skool.

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