library.onepin.app/epicatechin Peptide Education Library
Education only, not medical advice 21+ Every dose is an example to finalize with a licensed provider

OnePin Peptide Library · Metabolic

Metabolic Supplement Not FDA-approved · investigational Controlled substance

Epicatechin

(-)-Epicatechin

SupplementFlavonoid

Epicatechin (specifically (-)-epicatechin) is a naturally occurring flavanol found in high concentrations in dark chocolate (cacao), green tea, apples, and certain berries. It belongs to the flavan-3-ol subclass of flavonoids and has gained research interest for its potential effects on skeletal muscle physiology, cardiovascular health, and exercise performance. Epicatechin has been studied as a natural myostatin inhibitor and follistatin promoter, which has attracted attention in the sports nutrition and muscle-building communities.,Research, primarily from the laboratory of Dr. Francisco Villarreal at UC San Diego, has shown that epicatechin can modulate the myostatin-follistatin ratio in both animal models and small human studies. Myostatin is a negative regulator of muscle growth, and reducing its activity or increasing follistatin (which binds and inhibits myostatin) may promote muscle hypertrophy and improved muscle function. Additionally, epicatechin has demonstrated effects on mitochondrial biogenesis, nitric oxide production, and endothelial function.,Epicatechin is available as an over-the-counter dietary supplement and is generally recognized as safe (GRAS) as a food component. Clinical evidence for its muscle-building and performance-enhancing effects in humans remains preliminary, with most studies being small and short-term. Its cardiovascular benefits through nitric oxide-mediated vasodilation are better established in the broader flavanol literature.

Quick Start
Route
Oral
Start low
100-200mg
Frequency
daily
Timing
Can be taken with or without food. Some evidence suggests better absorption with a small amount of fat.

Start here. Every protocol below is ordered lowest-first. Begin at the smallest effective dose, hold about a week to assess tolerance, and step up only if needed.

Tiered Protocols · lowest first
Quick Start
Conservative start
100-200mg · Oral · daily
Lowest starting point. Hold about a week to assess tolerance before stepping up.
100-200mg
daily
Intermediate
Myostatin Inhibition
250-500 mg · Oral · Daily
human study · Gutierrez-Salmean et al. 2014 (J Nutr Biochem)
250-500 mg
Daily
Reconstitution CalculatorU-100
050100u
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units
01

How it works

Decreases myostatin and increases follistatin expression in skeletal muscle, shifting the balance toward a pro-anabolic signaling environment. This effect is mediated in part through modulation of the TGF-beta/Smad signaling pathway.,Stimulates mitochondrial biogenesis through activation of PGC-1alpha and SIRT1 pathways, increasing mitochondrial volume and oxidative capacity in muscle fibers. This may improve endurance and muscle fatigue resistance.,Enhances nitric oxide (NO) bioavailability by stimulating endothelial nitric oxide synthase (eNOS) activity, leading to improved vasodilation, blood flow, and reduced blood pressure. Also exerts antioxidant effects by scavenging reactive oxygen species.

Decreases myostatin and increases follistatin expression in skeletal muscle, shifting the balance toward a pro-anabolic signaling environment. This effect is mediated in part through modulation of the TGF-beta/Smad signaling pathway.,Stimulates mitochondrial biogenesis through activation of PGC-1alpha and SIRT1 pathways, increasing mitochondrial volume and oxidative capacity in muscle fibers. This may improve endurance and muscle fatigue resistance.,Enhances nitric oxide (NO) bioavailability by stimulating endothelial nitric oxide synthase (eNOS) activity, leading to improved vasodilation, blood flow, and reduced blood pressure. Also exerts antioxidant effects by scavenging reactive oxygen species.

02

What to expect

Early
Days 1–7

Days 1-7: Myostatin/follistatin ratio shifts detectable in blood work within 7 days (per published data at 1mg/kg/day). Nitric oxide effects may improve exercise performance subtly.

03

Evidence

HumanPresent
AnimalPresent
In-vitroPresent
2019Acute study of dose-dependent effects of (-)-epicatechin on vascular function in healthy male volunteers: A randomized controlled trial · Dower JI, Geleijnse JM, Hollman PC, et al, Clinical Nutrition ↗peer reviewed
2011(-)-Epicatechin enhances fatigue resistance and oxidative capacity in mouse muscle · Nogueira L, Ramirez-Sanchez I, Perkins GA, et al, Journal of Physiology ↗peer reviewed
2014Effects of (-)-epicatechin on molecular modulators of skeletal muscle growth and differentiation · Gutierrez-Salmean G, Ciaraldi TP, Nogueira L, et al, Journal of Nutritional Biochemistry ↗peer reviewed
2024Cocoa flavanols, Nrf2 activation, and oxidative stress in peripheral artery disease: mechanistic findings in muscle based on outcomes from a randomized trial · Komosinska-Vassev K, McDermott MM, Sufit RL, et al, American Journal of Physiology - Cell Physiology ↗peer reviewed
04

Interactions & stacking

What's safe to combine, and what belongs in a separate pin.

Safe & synergistic

BPC-157No pharmacological conflict - epicatechin supports muscle physiology while BPC-157 promotes tissue healing
Testosterone CypionateEpicatechin's myostatin inhibition may complement anabolic hormone effects on muscle growth
EnclomipheneNo interaction - independent mechanisms for muscle and hormonal support
NAD+Both support mitochondrial function through complementary pathways

Keep separate

Blood thinners (Warfarin)Flavonoids have mild antiplatelet activity - may potentiate anticoagulant effects and increase bleeding risk
05

Pharmacokinetics

Illustrative plasma concentration · 24 h
Half-life
~2-3 hours
Peak · Tmax
~1-2 hours oral
Elimination
~10-15 hours
Activity
6-12 hours (myostatin/follistatin ratio changes and NO enhancement persist beyond parent compound clearance)

Storage. Store in a cool, dry place away from light. Oral compound - no reconstitution needed. Some formulations recommend refrigeration.

06

Regulatory status

Dietary supplement (OTC) in the United States. Classified as a food component with GRAS status. Not FDA-approved as a drug for any indication. Not a controlled substance. Available worldwide as a nutritional supplement.

Put it to work

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Open Epicatechin straight into OnePin with your vial and dose pre-filled, then let it handle the syringe math and remind you before the vial runs out.

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The guide & community

The complete Epicatechin walkthrough, real protocol discussion and coaching live inside the BlessUp community on Skool.

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