library.onepin.app/ahk-cu Peptide Education Library
Education only, not medical advice 21+ Every dose is an example to finalize with a licensed provider

OnePin Peptide Library · Skin

Skin Copper-Bound Tripeptide Not FDA-approved · investigational

AHK-Cu

AHK Copper · Alanyl-Histidyl-Lysine Copper

Copper-Bound TripeptideHair Follicle StimulatorTopical CosmeceuticalResearch Chemical (no FDA approval)

AHK-Cu (Alanyl-Histidyl-Lysine-Copper) is a copper-bound tripeptide closely related to GHK-Cu. Where GHK-Cu primarily targets skin remodeling and collagen biology, AHK-Cu is more specifically researched for hair follicle stimulation and hair regrowth. The copper coordination chemistry and downstream signaling overlap substantially with GHK-Cu - both peptides bind copper(II) in a 1:1 complex and modulate gene expression related to extracellular matrix remodeling, angiogenesis, and antioxidant defense.

Quick Start
Route
Topical (only defensible route; injecting AHK-Cu is not advised - no injectable data)
Start low
1-3% topical serum/solution (start 0.5%, step to 1-2% if tolerated)
Frequency
Daily topical / 1-2x weekly injection
Timing
Independent

Topical: apply to scalp daily, leave on overnight. Injectable: 1-2x weekly to scalp area. Light-sensitive (copper complex).

Start here. Every protocol below is ordered lowest-first. Begin at the smallest effective dose, hold about a week to assess tolerance, and step up only if needed.

Tiered Protocols · lowest first
Quick Start
Conservative start
1-3% topical serum/solution (start 0.5%, step to 1-2% if tolerated) · Topical (only defensible route; injecting AHK-Cu is not advised - no injectable data) · Daily topical / 1-2x weekly injection
Lowest starting point. Hold about a week to assess tolerance before stepping up.
1-3% topical serum/solution (start 0.5%, step to 1-2% if tolerated)
Daily topical / 1-2x weekly injection
Standard
Hair Follicle Stimulation
3-5 % · Topical · Daily
in vitro · Pyo et al. 2007 (Arch Pharm Res)
3-5 %
Daily
Reconstitution CalculatorU-100
050100u
Draw to
units
01

How it works

AHK-Cu chelates copper(II) in 1:1 stoichiometry, similar to GHK-Cu. The peptide-copper complex is taken up by cells via reduction at the membrane and modulates intracellular gene expression:

Hair Follicle Stimulation

Promotes vellus-to-terminal hair conversion in dermal papilla cell cultures. Upregulates VEGF, FGF-7 (KGF), and other growth factors at hair follicles.

Copper Coordination

Same coordination chemistry as GHK-Cu - copper conjugation is the bioactive form. Copper-free forms have reduced or absent activity.

Same Chemistry Conflicts as GHK-Cu

NEVER co-store with thiol/Met/Cys-containing peptides. Copper drives oxidation of these residues during co-storage, degrading both peptides.

Topical Penetration

Small tripeptide passes through stratum corneum reasonably well. Often formulated with penetration enhancers in commercial products.

Synergy with GHK-Cu

Often combined - GHK-Cu for skin/scalp matrix, AHK-Cu for hair-specific follicle stimulation.

02

What to expect

Early
Days 1–7

Weeks 1-4: minimal subjective change.

Mid
Weeks 2–4

Weeks 4-12: subtle hair texture improvements.

Later
Weeks 4–12

Weeks 12-24: visible hair density increase if responsive.

03

Evidence

HumanModerate
AnimalPresent
In-vitroPresent
2018Tripeptide-copper complexes for skin and hair regeneration · Pickart L, Margolina A, International Journal of Molecular Sciences ↗review
1993Effect of copper tripeptide on hair growth in mice · Uno H, Kurata S, Skin Pharmacology ↗peer reviewed
2008Use of tricopeptides for the treatment of hair loss · Pickart L, Cosmetics & Toiletries ↗review
04

Interactions & stacking

What's safe to combine, and what belongs in a separate pin.

Keep separate

05

Side effects & safety

Commonly reported

  • Mild scalp irritation (topical)
  • Mild injection site reaction (injectable)
  • Temporary scalp redness

Less common & notes

  • Allergic reaction to peptide or formulation.
  • Copper-related effects rare with topical use due to low systemic absorption.
  • Injectable use carries the standard copper-peptide chemistry concerns.
06

Pharmacokinetics

Illustrative plasma concentration · 24 h
Half-life
Hours plasma; tissue effects days-weeks
Peak · Tmax
Topical 30-60 min, SubQ 1-2 hours
Elimination
Hours plasma; hair effects accumulate over weeks
Activity
Hair effects build over 12-24 weeks

Storage. Refrigerate. Light-sensitive (copper complex). Reconstituted: 21-28 days refrigerated. Discard if color changes.

07

Regulatory status

Not FDA-approved. Sold as cosmeceutical (topical) or research chemical (injectable). WADA: not specifically prohibited.

Put it to work

Calculate, log & track

Open AHK-Cu straight into OnePin with your vial and dose pre-filled, then let it handle the syringe math and remind you before the vial runs out.

Open AHK-Cu in the app →

Go deeper

The guide & community

The complete AHK-Cu walkthrough, real protocol discussion and coaching live inside the BlessUp community on Skool.

Join the community ↗
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